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Pile Of Books

PUBLICATIONS

Publications: List

h-index of 18, total citations >1200

  1. Modha, Sachin G.; Pöthig, Alexander; Dreuw, Andreas; Bach, Thorsten.* “[6π] Photocyclization to cis-Hexahydrocarbazol-4-ones: Substrate modification, mechanism and scope” J. Org. Chem. 2019, 84, 1139-1153. (Selected as Featured Article)  https://pubs.acs.org/doi/abs/10.1021/acs.joc.8b03144

  2. Modha, Sachin G.; Popescu, Mihai V.; Greaney, Michael F.* “Synthesis of Triarylamines via sequential C-N bond formation” J. Org. Chem. 2017, 82, 11933-11938. (Invited article for a special issue on hypervalent iodine chemistry)  https://pubs.acs.org/doi/abs/10.1021/acs.joc.7b01778

  3. Teskey, Christopher J.; Sohel, Shariar M. A.; Bunting, Danielle L.; Modha, Sachin G.; Greaney, Michael F.* “Domino N-/C-Arylation via in situ generation of a directing group: Atom-Efficient Arylation uding diaryliodonium salts” Angew. Chem. Int. Ed., 2017, 56, 5263-5266. (This paper is selected as Hot Paper by the Journal) https://onlinelibrary.wiley.com/doi/10.1002/anie.201701523

  4. Modha, Sachin G.; Greaney, Michael F.* “Atom-economical transformations of diaryliodonium salts: Tandem C-H and N-H arylation of indoles” J. Am. Chem. Soc., 2015, 137, 1416-1419. (Featured in Chemical and Engineering News)  https://pubs.acs.org/doi/10.1021/ja5124754

  5. Vachhani, Dipak D.; Kumar, Amit; Modha, Sachin G.;* Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V.* “Diversely substituted indoloazepinones and indoloazocinones: A post-Ugi Gold-catalyzed regioselective carbocyclization approach” Synthesis, 2015, 47, 1337-1347.  https://www.thieme-connect.com/products/ejournals/abstract/10.1055/s-0034-1379894

  6. Modha, Sachin G.; Van der Eycken, Erik V. “Reactions with [3+2] cycloaddition as the key step” In Science of Synthesis: Multicomponent Reactions, Muller, T. J. J., Ed.; Thieme: Stuttgart, (2014), Vol. 2, pp 287-302. ISBN: 9783131728517.

  7. Kumar, Amit; Vachhani, Dipak D.; Modha, Sachin G.;* Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V.* “Post-Ugi Gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines” Beilstein J. Org. Chem., 2013, 9, 2097-2102.  https://www.beilstein-journals.org/bjoc/articles/1860-5397-9-246

  8. Kumar, Amit; Vachhani, Dipak D.; Modha, Sachin G.;* Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V.* “Post Ugi Gold(I)- and Platinum(II)-catalyzed alkyne activation: Synthesis of diversely substituted fused azepinones and pyridinones” Synthesis, 2013, 45, 2571-2582. https://www.thieme-connect.com/products/ejournals/abstract/10.1055/s-0033-1339474

  9. Modha, Sachin G.; Mehta, Vaibhav P.; Van der Eycken, Erik V.* “Transition metal-catalyzed C-C bond formation via C-S bond cleavage: an overview” Chem. Soc. Rev., 2013, 42, 5042-5055. https://pubs.rsc.org/en/content/articlelanding/2013/cs/c3cs60041f/unauth#!divAbstract

  10. Kumar, Amit; Vachhani, Dipak D.; Modha, Sachin G.; Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V. “Gold(I)-catalyzed post-Ugi hydroarylation: An approach to pyrrolopyridines and azepinoindoles” Eur. J. Org. Chem., 2013, 2288-2292.*

  11. Vachhani, Dipak D.; Kumar, Amit; Modha, Sachin G.; Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V. “Diversely substituted triazolo[1,5-a][1,4]benzodiazepinones: A post-Ugi Copper-catalyzed tandem azide-alkyne cycloaddition/Ullmann C-N coupling approach” Eur. J. Org. Chem., 2013, 1223-1227.

  12. Vachhani, Dipak D.; Modha, Sachin G.; Sharma, Abhishek; Van der Eycken, Erik V. “A facile diversity-oriented synthesis of imidazo[1,2-a]pyrazinones via Gold-catalyzed regioselective heteroannuation of propynylaminopyrazinones” Tetrahedron, 2013, 69, 359-365.

  13. Mishra, Nigam M.; Vachhani, Dipak D.; Modha, Sachin G.; Van der Eycken, Erik V. “Diversely substituted imidazo[1,2-a]pyrazine-8-oxo-3-carbaldehydes: An iodine-mediated cyclization/oxidation approach” Eur. J. Org. Chem. 2013, 693-700.

  14. Modha, Sachin G.; Kumar, Amit; Vachhani, Dipak D.; Sharma, Sunil K.; Parmar, Virinder S.; Van der Eycken, Erik V. “Gold(I) and Platinum(II) switch: a post-Ugi intramolecular hydroarylation to pyrrolopyridinones and pyrroloazepinones” Chem. Commun., 2012, 48, 10916-10918.

  15. Modha, Sachin G.; Kumar, Amit; Vachhani, Dipak D.; Jacobs, Jeroen; Sharma, Sunil K.; Parmar, Virinder S.; Van Meervelt, Luc; Van der Eycken, Erik V. “A diversity-oriented approach to spiroindolines: Post-Ugi Gold-catalyzed diastereoselective domino cyclization” Angew. Chem. Int. Ed., 2012, 51, 9572-9575.

  16. Mishra, Nigam M.; Peshkov, Vsevolod A.; Pereshivko, Olga P.; Modha, Sachin G.; Van der Eycken, Erik V. “Alkylation of 3,5-dichloro-2(1H)-pyrazinones using malonate esters” Tetrahedron Lett., 2012, 53, 4676-4678.

  17. Modha, Sachin G.; Vachhani, Dipak D.; Jacobs, Jeroen; Van Meervelt, Luc; Van der Eycken, Erik V. “A concise route to indoloazocines via a sequential Ugi-Gold-catalyzed intramolecular hydroarylation” Chem. Commun. 2012, 48, 6550-6552. (Listed by Synfacts DOI: 10.1055/s-0032-1316700).

  18. Modha, Sachin G.; Trivedi, Jalpa C.; Mehta, Vaibhav P.; Ermolat’ev, Denis S.; Van der Eycken, Erik V. “Efficient preparation of tetrasubstituted pyrazines starting from pyrazine-2(1H)-ones” Synthesis, 2012, 44, 1614-1624.

  19. Vachhani, Dipak D.; Mehta, Vaibhav P.; Modha, Sachin G.; Van Hecke, Kristof; Van Meervelt, Luc; Van der Eycken, Erik V. “Microwave-assisted synthesis of pyrazino[2,1-b]quinazolines and 3-indolyl-2(1H)-pyrazinones employing a chemoselective Silver(I)- and Gold(I)-catalyzed reaction” Adv. Synth. Catal., 2012, 354, 1593-1599.

  20. Mehta, Vaibhav P.; Modha, Sachin G.; Ruijter, Eilco; Van Hecke, Kristof; Van Meervelt, Luc; Pannecouque, Christophe; Balzarini, Jan; Orru, Romano V. A.; Van der Eycken, Erik “A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: Synthesis and biological evaluation” J. Org. Chem., 2011, 76(8), 2828-2839. (Listed by Synfacts DOI: 10.1055/s-0030-1260688).

  21. Mehta, Vaibhav P.; Sharma, Ajendra K.; Modha, Sachin G.; Sharma, Sweta; Meganathan, Thirumal; Parmar, Virinder S.; Van der Eycken, Erik “N-Heterocyclic carbene catalyzed aroylation of 3,5-dichloro-2(1H)-pyrazinones” J. Org. Chem., 2011, 76(8), 2920-2925.

  22. Modha, Sachin G.; Trivedi, Jalpa C.; Mehta, Vaibhav P.; Ermolat’ev, Denis S.; Van der Eycken, Erik V. “An expeditious route toward pyrazine-containing nucleoside analogues” J. Org. Chem. 2011, 76(3), 846-856.

  23. Mehta, Vaibhav P.; Modha, Sachin G.; Van der Eycken, Erik V. “Microwave-assisted Palladium-catalyzed phosphonium coupling of 2(1H)-pyrazinones” J. Org. Chem., 2010, 75, 976-979.

  24. Modha, Sachin G.; Mehta, Vaibhav P.; Ermolat’ev, Denis; Balzarini, Jan; Van Hecke, Kristof ; Van Meervelt, Luc; Van der Eycken, Erik V. “Microwave-assisted synthesis of a novel class of imidazolylthiazolidin-4-ones and evaluation of its biological activities”  Mol. Divers., 2010, 14(4), 767-776.

  25. Van Overschelde, Michel; Vervecken, Elias; Modha, Sachin G.; Cogen, Simon; Van der Eycken, Erik; Van der Eycken, Johan “Catalyst-free alcoholysis of phosphane-boranes: a smooth, cheap, and efficient deprotection procedure” Tetrahedron, 2009, 65(32), 6410-6415.

  26. Francois, Isabelle E. J. A.; Cammue, Bruno P. A.; Bresseleers, Sara; Fleuren, Hein; Hoornaert, Georges; Mehta, Vaibhav P.; Modha, Sachin G.; Van der Eycken, Erik V.; Thevissen, Karin “Synthesis and fungicidal activity of 3,5-dichloropyrazine-2(1H)-one derivatives” Bioorg. Med. Chem. Lett., 2009, 19(15), 4064-4066.

  27. Mehta, Vaibhav P.; Modha, Sachin G.; Ermolat'ev, Denis; Van Hecke, Kristof; Van Meervelt, Luc; Van der Eycken, Erik V. “Diversity-oriented synthesis of substituted furo[2,3-b]pyrazines” Aust. J. Chem., 2009, 62(1), 27-41.

  28. Mehta, Vaibhav P.; Modha, Sachin G.; Van der Eycken, Erik “Mild room-temperature Palladium-catalyzed C3-arylation of 2(1H)-pyrazinones via a desulfitative kumada-type cross-coupling reaction” J. Org. Chem. 2009, 74(17), 6870-6873.

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